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+27 31 260 7358
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Dr. Rajshekhar Karpoormath

Person

     Dr Rajshekhar Karpoormath

Telephone

+27 (0) 31 260 7179

Email

karpoormath@ukzn.ac.za 

Campus

Westville

Designation

Senior Lecturer

Research Interests

  • Target based Drug design and Synthesis 
  • Organic Synthesis and Methodology development Biosensors

List of Publications

  1. Rajshekhar Karpoormath, Fernando Albericio, Thavendran Govender, GlennE M. Maguire and HendrikG Kruger, 'Synthesis and NMR elucidation of pentacycloundecane-derived hydroxy acid peptides as potential anti-HIV-1 agents', Structural Chemistry,2013 (In Press), pp. 1-11.
  2. Rajshekhar Karpoormath, Yasien Sayed, Thavendran Govender, Hendrik G. Kruger, Mahmoud E. S. Soliman and Glenn E. M. Maguire, 'Novel PCU cage diol peptides as potential targets against wild-type CSA HIV-1 protease: synthesis, biological screening and molecular modelling studies', Medicinal Chemistry Research, 2013 (In Press), p. Ahead of Print.
  3. Rajshekhar Karpoormath, Oluseye K. Onajole, Tricia Naicker, Thavendran Govender, Glenn E. M. Maguire and Hendrik G. Kruger, 'Synthesis and NMR elucidation of novel pentacycloundecane-derived peptides', South African Journal of Chemistry, Vol. 65, 2012, pp. 108-14.
  4. Rajshekhar Karpoormath, Yasien Sayed, Patrick Govender, Thavendran Govender, Hendrik G. Kruger, Mahmoud E. S. Soliman and Glenn E. M. Maguire, 'Pentacycloundecane derived hydroxy acid peptides: A new class of irreversible non-scissile ether bridged type isoster as potential HIV-1 wild type C-SA protease inhibitors', Bioorganic Chemistry, Vol. 40, Feb 2012, pp. 19-29.
  5. Rajshekhar Karpoormath, Patrick Govender, Thavendran Govender, Hendrik G. Kruger and Glenn E. M. Maguire, 'endo-11-(Dibenzylamino)tetracyclo[5.4.0.0(3,10).0(5,9)]undecane-8-one', Acta Crystallographica Section E-Structure Reports Online, Vol. 67, Mar 2011, pp. O619-U1716.
  6. Rajshekhar Karpoormath, Tricia Naicker, Thavendran Govender, Hendrik G. Kruger and Glenn E. M. Maguire, 'Benzyl 5-hydroxy-4-oxapentacyclo[5.4.1.02,6.03,10.08,11]dodecane-3-carboxylate', Acta Crystallographica Section E-Structure Reports Online, Vol. 67, Apr 2011, pp. O877-U539.
  7. Rajshekhar Karpoormath, Patrick Govender, Hendrik G. Kruger, Thavendran Govender and Glenn E. M. Maguire, 'N,N '-[(8-endo,11-endo-Dihydroxypentacyclo[5.4.0.0(2,6).0(3,10).0(5,9)]undec ane-8,11-diyl)bis(methylenecarbonyl)]di-L-phenylalanine', Acta Crystallographica Section E-Structure Reports Online, Vol. 66, Oct 2010, pp. O2537-U268.
  8. Rajshekhar Karpoormath, Thavendran Govender, Patrick Govender, Hendrik G. Kruger and Glenn E. M. Maguire, 'tert-Butyl N-[(11-exo-benzyloxycarbonyl-8-oxopentacyclo[5.4.0.0(2,6).0(3,10).0(5,9) ]undecane-11-endo-yloxy)carbonyl-methyl] carbamate', Acta Crystallographica Section E-Structure Reports Online, Vol. 66, Oct 2010, pp. O2607-U900.
  9. Grant A. Boyle, Thavendran Govender, Rajshekhar Karpoormath and Hendrik G. Kruger, 'exo-8,exo-11-Diallylpentacyclo-[5.4.0.0(2,6).0(3,10).0(5,9)]undecane-end o-8,endo-11-diol', Acta Crystallographica Section E-Structure Reports Online, Vol. 63, Dec2007, pp. O4797-U5875.
  10. Grant A. Boyle, Thavendran Govender, Rajshekhar Karpoormath and Hendrik G. Kruger, 'exo-8,exo-11-Divinylpentacyclo[5.4.0.0(2,6).0(3,10).0(5,6)]undecane-endo -8, endo-11-diol', Acta Crystallographica Section E-Structure Reports Online, Vol. 63, Oct2007, pp. O3977-U2352.
  11. K. Gadad, M. N. Noolvi and R. V. Karpoormath, 'Synthesis and anti-tubercular activity of a series of 2-sulfonamido/trifluoromethyl-6-substituted imidazo[2,1-b]-1,3,4-thiadiazole derivatives', Bioorganic & Medicinal Chemistry, Vol. 12, no. 21, Nov 1 2004, pp. 5651-9.
 

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